A Combinatorial Approach to [1,5]Benzothiazepine Derivatives as Potential Antibacterial Agents
Journal of Combinatorial Chemistry2001Vol. 3(2), pp. 224–228
Citations Over TimeTop 25% of 2001 papers
Fabrizio Micheli, Fabio Degiorgis, Aldo Feriani, Alfredo Paio, Alfonso Pozzan, Paola Zarantonello, Pierfausto Seneci
Abstract
[1,5]Benzothiazepines are widely used in a number of different therapeutic areas and therefore represent an interesting scaffold for de novo exploration. Recent literature reports suggest their value as antibacterial agents. The present paper reports the exploration of this scaffold for the generation of combinatorial libraries both in solution and on solid phase.
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