De Novo Design of a Novel Oxazolidinone Analogue as a Potent and Selective α1A Adrenergic Receptor Antagonist with High Oral Bioavailability
Citations Over TimeTop 15% of 2000 papers
Abstract
ADVERTISEMENT RETURN TO ISSUELetterNEXTDe Novo Design of a Novel Oxazolidinone Analogue as a Potent and Selective α1A Adrenergic Receptor Antagonist with High Oral BioavailabilityBharat Lagu, Dake Tian, Yoon Jeon, Chao Li, John M. Wetzel, Dhanapalan Nagarathnam, Quanrong Shen, Carlos Forray, Raymond S. L. Chang, Theodore P. Broten, Richard W. Ransom, Tsing-Bao Chan, Stacey S. O'Malley, Terry W. Schorn, A. David Rodrigues, Kelem Kassahun, Douglas J. Pettibone, Roger Freidinger, and Charles GluchowskiView Author Information Departments of Chemistry and Pharmacology, Synaptic Pharmaceutical Corporation, 215 College Road, Paramus, New Jersey 07652, and Departments of Medicinal Chemistry, Pharmacology, and Drug Metabolism, Merck Research Laboratories, West Point, Pennsylvania 19486 Cite this: J. Med. Chem. 2000, 43, 15, 2775–2778Publication Date (Web):July 7, 2000Publication History Received25 February 2000Published online7 July 2000Published inissue 1 July 2000https://pubs.acs.org/doi/10.1021/jm000085ehttps://doi.org/10.1021/jm000085erapid-communicationACS PublicationsCopyright © 2000 American Chemical SocietyRequest reuse permissionsArticle Views595Altmetric-Citations17LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InRedditEmail Other access optionsGet e-AlertscloseSupporting Info (1)»Supporting Information Supporting Information SUBJECTS:Anatomy,Antagonists,Receptors,Rodent models,Screening assays Get e-Alerts
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