Copper-catalyzed annulation of amidines for quinazoline synthesis
Chemical Communications2013Vol. 49(57), pp. 6439–6439
Citations Over TimeTop 10% of 2013 papers
Abstract
An efficient Cu-catalyzed synthesis of quinazolines via the C-N bond formation reactions between N-H bonds of amidines and C(sp(3))-H bonds adjacent to sulfur or nitrogen atoms in the commonly used solvents, such as DMSO, DMF, DMA, NMP or TMEDA, followed by intramolecular C-C bond formation reactions was developed for the first time.
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