Antagonism of the proinflammatory and pronociceptive actions of canonical and biased agonists of protease‐activated receptor‐2
British Journal of Pharmacology2016Vol. 173(18), pp. 2752–2765
Citations Over TimeTop 22% of 2016 papers
TinaMarie Lieu, Emilia E. Savage, Peishen Zhao, Laura E. Edgington‐Mitchell, Νicholas Barlow, Romke Bron, Daniel P. Poole, Peter McLean, Rink‐Jan Lohman, David P. Fairlie, Nigel W. Bunnett
Abstract
GB88 inhibits the capacity of canonical and biased protease agonists of PAR2 to cause nociception and inflammation.
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