Jyothi Mahadevaswamy
AstraZeneca (India)(IN)
Publications by Year
Research Areas
Biochemical and Molecular Research, Tuberculosis Research and Epidemiology, Cancer therapeutics and mechanisms, Synthesis and biological activity, HIV/AIDS drug development and treatment
Most-Cited Works
- → Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious in Vivo(2013)161 cited
- → 4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity(2014)94 cited
- → Discovery of Pyrazolopyridones as a Novel Class of Noncovalent DprE1 Inhibitor with Potent Anti-Mycobacterial Activity(2014)93 cited
- → Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase(2015)58 cited
- → Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial Activity(2019)40 cited
- Discovery of benzothiazoles as antimycobacterial agents: synthesis, structure-activity relationships and binding studies with<em> </em>Mycobacterium tuberculosis<em> </em>decaprenylphosphoryl-β-d-ribose 2′-oxidase(2015)