Kaustav Biswas
Merck & Co., Inc., Rahway, NJ, USA (United States)(US)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Coagulation, Bradykinin, Polyphosphates, and Angioedema, Synthetic Organic Chemistry Methods, Cancer Treatment and Pharmacology, Neuropeptides and Animal Physiology
Most-Cited Works
- → Parallel Synthesis and Screening of a Solid Phase Carbohydrate Library(1996)278 cited
- → Highly Concise Routes to Epothilones: The Total Synthesis and Evaluation of Epothilone 490(2002)111 cited
- → Unfolded Protein Response in Cancer: IRE1α Inhibition by Selective Kinase Ligands Does Not Impair Tumor Cell Viability(2014)104 cited
- → Effects of temperature and concentration in some ring closing metathesis reactions(2003)68 cited
- → Discovery of TRPM8 Antagonist (S)-6-(((3-Fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamoyl)nicotinic Acid (AMG 333), a Clinical Candidate for the Treatment of Migraine(2018)61 cited
- → NanoClick: A High Throughput, Target-Agnostic Peptide Cell Permeability Assay(2021)58 cited
- → Application of hitherto unexplored macrocyclization strategies in the epothilone series: novel epothilone analogs by total synthesisElectronic supplementary information (ESI) available: experimental details for the synthesis of 14 and 32. See http://www.rsc.org/suppdata/cc/b2/b209941a/(2002)55 cited
- → Single Residue Substitutions That Confer Voltage-Gated Sodium Ion Channel Subtype Selectivity in the NaV1.7 Inhibitory Peptide GpTx-1(2016)51 cited
- → Total Syntheses of [17]- and [18]Dehydrodesoxyepothilones B via a Concise Ring-Closing Metathesis-Based Strategy: Correlation of Ring Size with Biological Activity in the Epothilone Series(2002)50 cited
- → Pharmacological characterization of potent and selective NaV1.7 inhibitors engineered from Chilobrachys jingzhao tarantula venom peptide JzTx-V(2018)49 cited