Thomas E. Rawson
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Cancer-related Molecular Pathways, Synthesis and Characterization of Heterocyclic Compounds, Protein Kinase Regulation and GTPase Signaling, Computational Drug Discovery Methods
Most-Cited Works
- → Benzodiazepine Peptidomimetics: Potent Inhibitors of Ras Farnesylation In Animal Cells(1993)628 cited
- → From Peptide to Non-Peptide. 2. The de Novo Design of Potent, Non-peptidal Inhibitors of Platelet Aggregation Based on a Benzodiazepinedione Scaffold(1994)99 cited
- → A Class of 2,4-Bisanilinopyrimidine Aurora A Inhibitors with Unusually High Selectivity against Aurora B(2009)81 cited
- → Potent α4β1 Peptide Antagonists as Potential Anti-Inflammatory Agents(1997)80 cited
- → In vitro characterization of four novel classes of growth hormone-releasing peptide.(1995)66 cited
- → A Pentacyclic Aurora Kinase Inhibitor (AKI-001) with High in Vivo Potency and Oral Bioavailability(2008)58 cited
- → Benzodiazepine peptidomimetic inhibitors of farnesyltransferase(1994)51 cited
- → A Selective, Slow Binding Inhibitor of Factor VIIa Binds to a Nonstandard Active Site Conformation and Attenuates Thrombus Formation in Vivo(2005)41 cited
- → Separation of 21 -(R)- and 21-(S)-Argatroban: Solubility and Activity of the Individual Diastereoisomers(1993)15 cited
- → The synthesis of chiral 3-oxo-6-[(phenylmethoxy)-carbonyl]-2-piperazineacetic acid esters designed for the presentation of an aspartic acid side chain. A subsequent novel Friedel Crafts reaction(1992)15 cited