Yasunori Hase
Publications by Year
Research Areas
Synthesis and Biological Evaluation, Synthesis and Catalytic Reactions, Asymmetric Synthesis and Catalysis, Psoriasis: Treatment and Pathogenesis, Blood Coagulation and Thrombosis Mechanisms
Most-Cited Works
- → Catalytic Asymmetric Aminolysis of 3,5,8-Trioxabicyclo[5.1.0]octane Providing an Optically Pure 2-Amino-1,3,4-butanetriol Equivalent(1999)139 cited
- → Discovery of Conformationally Constrained Tetracyclic Compounds as Potent Hepatitis C Virus NS5B RNA Polymerase Inhibitors(2006)111 cited
- → SAR Exploration Guided by LE and Fsp 3 : Discovery of a Selective and Orally Efficacious RORγ Inhibitor(2015)58 cited
- → Discovery of a Janus Kinase Inhibitor Bearing a Highly Three-Dimensional Spiro Scaffold: JTE-052 (Delgocitinib) as a New Dermatological Agent to Treat Inflammatory Skin Disorders(2020)52 cited
- → Discovery of JTZ-951: A HIF Prolyl Hydroxylase Inhibitor for the Treatment of Renal Anemia(2017)51 cited
- → Discovery of (1S,2R,3R)-2,3-Dimethyl-2-phenyl-1-sulfamidocyclopropanecarboxylates: Novel and Highly Selective Aggrecanase Inhibitors(2011)49 cited
- → Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCβ-selective inhibitors(2006)44 cited
- → Discovery of Second Generation RORγ Inhibitors Composed of an Azole Scaffold(2019)31 cited
- → Synthesis and Structure−Activity Relationships of 5,6,7,8-Tetrahydro-4H-thieno[3,2-b]azepine Derivatives: Novel Arginine Vasopressin Antagonists(2003)27 cited
- → Synthesis and Structure−Activity Relationships of Novel Selective Factor Xa Inhibitors with a Tetrahydroisoquinoline Ring(2005)22 cited