Prakash Vachaspati
Syngene International (India)(IN)
Publications by Year
Research Areas
Cancer therapeutics and mechanisms, Biochemical and Molecular Research, Pharmacogenetics and Drug Metabolism, Phenothiazines and Benzothiazines Synthesis and Activities, Tuberculosis Research and Epidemiology
Most-Cited Works
- → Thiazolopyridine Ureas as Novel Antitubercular Agents Acting through Inhibition of DNA Gyrase B(2013)66 cited
- → Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase(2015)58 cited
- → Diarylthiazole: An Antimycobacterial Scaffold Potentially Targeting PrrB-PrrA Two-Component System(2014)47 cited
- → Optimised method to estimate octanol water distribution coefficient (logD) in a high throughput format(2016)38 cited
- → Nitroarenes as Antitubercular Agents: Stereoelectronic Modulation to Mitigate Mutagenicity(2016)24 cited
- → The synthesis and evaluation of benzannelated-azatoxins: The benzazatoxins(1998)11 cited
- → A Proposed Mechanism for p-Aminoclonidine Allergenicity Based on Its Relative Oxidative Lability(1997)7 cited
- → Fast mouse PK (Fast PK): A rapid screening method to increase pharmacokinetic throughput in pre-clinical drug discovery(2012)7 cited
- → Beyond Bioisosteres: Impact of Replacing a Benzene Ring with sp 3 -Rich Three-Dimensional Saturated Bridged Bicyclic Match Pairs on Biotransformation, Metabolic Stability, and Other ADME Profiles(2025)4 cited
- → Identification and characterization of a novel ergothioneine conjugate of raloxifene(2025)2 cited