David G. Livermore

Publications by Year

Research Areas

Neuroendocrine regulation and behavior, Organic and Inorganic Chemical Reactions, Adenosine and Purinergic Signaling, Biochemical and Molecular Research, Synthesis and biological activity

Most-Cited Works

• → Discovery and structure–activity relationships of a series of pyroglutamic acid amide antagonists of the P2X7 receptor(2010)70 cited
• → 2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: identification, stereochemistry and initial SAR(2005)66 cited
• → Identification of regions of the P2X₇receptor that contribute to human and rat species differences in antagonist effects(2008)64 cited
• → 2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists. 2. Synthesis, Chirality, and Pharmacokinetics(2005)53 cited
• → 2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists. 3. Synthesis, Pharmacokinetics, and in Vivo Potency(2006)44 cited
• → Identification of potent and selective oxytocin antagonists. Part 2: further investigation of benzofuran derivatives(2002)42 cited
• → 1,2,4-Triazolo-[1,5-a]pyridine HIF Prolylhydroxylase Domain-1 (PHD-1) Inhibitors With a Novel Monodentate Binding Interaction(2017)33 cited
• → Identification of potent and selective oxytocin antagonists. Part 1: indole and benzofuran derivatives(2002)30 cited
• → Assessment of the Target Engagement and d-Serine Biomarker Profiles of the d-Amino Acid Oxidase Inhibitors Sodium Benzoate and PGM030756(2017)29 cited
• → Synthesis and structure–activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor(2010)27 cited