Jean-Michel Lefrançois
Galapagos (France)(FR)
Publications by Year
Research Areas
Estrogen and related hormone effects, Asymmetric Synthesis and Catalysis, Chemical Synthesis and Analysis, Cyclopropane Reaction Mechanisms, Coordination Chemistry and Organometallics
Most-Cited Works
- → Discovery and Optimization of an Azetidine Chemical Series As a Free Fatty Acid Receptor 2 (FFA2) Antagonist: From Hit to Clinic(2014)109 cited
- → Discovery of Diarylhydantoins as New Selective Androgen Receptor Modulators(2012)75 cited
- → Identification of a 4-(Hydroxymethyl)diarylhydantoin as a Selective Androgen Receptor Modulator(2012)51 cited
- → Diastereoselective Carbometalation of Vinyl Metals(1994)47 cited
- → Iodocyclization of olefinic t-butyl ethers : an easy stereocontrolled synthesis of cis-substituted tetrahydrofurans.(1992)39 cited
- → Acyclic stereocontrol through the metalla-claisen rearrangement. Part I(1991)26 cited
- → Acyclic Stereocontrol via Organogembismetallic Reagents; Part III1(1992)22 cited
- → Organobismetallic zinc reagents: Their preparation and use in diastereoselective reactions(1992)20 cited
- → Structure−Activity Relationships of a New Family of Steroidal Aromatase Inhibitors. 1. Synthesis and Evaluation of a Series of Analogs Related to 19-[(Methylthio)methyl]androstenedione (RU54115)(1996)18 cited
- → Biphenyls as Surrogates of the Steroidal Backbone. Part 2: Discovery of a Novel Family of Non-steroidal 5-α-Reductase Inhibitors(2001)12 cited