Pascal Heitel
Goethe University Frankfurt(DE)
Publications by Year
Research Areas
Peroxisome Proliferator-Activated Receptors, Drug Transport and Resistance Mechanisms, Estrogen and related hormone effects, Retinoids in leukemia and cellular processes, Computational Drug Discovery Methods
Most-Cited Works
- → Opportunities and Challenges for Fatty Acid Mimetics in Drug Discovery(2017)86 cited
- → Nonacidic Farnesoid X Receptor Modulators(2017)83 cited
- → DrugBank screening revealed alitretinoin and bexarotene as liver X receptor modulators(2017)52 cited
- → l-Thyroxin and the Nonclassical Thyroid Hormone TETRAC Are Potent Activators of PPARγ(2020)47 cited
- → Computer-Assisted Discovery and Structural Optimization of a Novel Retinoid X Receptor Agonist Chemotype(2019)43 cited
- → Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation(2023)42 cited
- → Boosting Anti-Inflammatory Potency of Zafirlukast by Designed Polypharmacology(2018)37 cited
- → Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain(2021)26 cited
- → Design and Structural Optimization of Dual FXR/PPARδ Activators(2020)26 cited
- → Emerging TACnology: Heterobifunctional Small Molecule Inducers of Targeted Posttranslational Protein Modifications(2023)21 cited