Daniel R. Gentile
Howard Hughes Medical Institute(US)University of California, San Francisco(US)
Publications by Year
Research Areas
Biochemical and Molecular Research, Protein Kinase Regulation and GTPase Signaling, Enzyme function and inhibition, Inflammatory mediators and NSAID effects, Monoclonal and Polyclonal Antibodies Research
Most-Cited Works
- → Aspirin’s Active Metabolite Salicylic Acid Targets High Mobility Group Box 1 to Modulate Inflammatory Responses(2015)119 cited
- → Ras Binder Induces a Modified Switch-II Pocket in GTP and GDP States(2017)116 cited
- → Novel K-Ras G12C Switch-II Covalent Binders Destabilize Ras and Accelerate Nucleotide Exchange(2018)61 cited
- Development of Second Generation Ras Switch-II Pocket Inhibitors(2017)