Eric Haaksma
Publications by Year
Research Areas
Receptor Mechanisms and Signaling, Chemical Synthesis and Analysis, Mast cells and histamine, Computational Drug Discovery Methods, Drug Transport and Resistance Mechanisms
Most-Cited Works
- → Target Binding Properties and Cellular Activity of Afatinib (BIBW 2992), an Irreversible ErbB Family Blocker(2012)858 cited
- → Ligand efficiency as a guide in fragment hit selection and optimization(2010)244 cited
- → Serine and Threonine Residues Bend α-Helices in the χ1=g− Conformation(2000)184 cited
- → GRID/CPCA: A New Computational Tool To Design Selective Ligands(2000)184 cited
- → Linking agonist binding to histamine H1 receptor activation(2005)93 cited
- → Discovery of Quinazolines as Histamine H4Receptor Inverse Agonists Using a Scaffold Hopping Approach(2008)88 cited
- → Histamine receptors: subclasses and specific ligands(1990)82 cited
- → Delineation of Agonist Binding to the Human Histamine H4Receptor Using Mutational Analysis, Homology Modeling, and ab Initio Calculations(2008)58 cited
- → In silicoprediction of substrate properties for ABC-multidrug transporters(2008)46 cited
- → Predicting Ligand Interactions with ABC Transporters in ADME(2009)45 cited