George B. Hill

Publications by Year

Research Areas

Microtubule and mitosis dynamics, Cancer-related Molecular Pathways, Synthesis and Biological Evaluation, Synthesis and Reactivity of Heterocycles, Synthesis and biological activity

Most-Cited Works

• → Discovery of a Potent and Selective EGFR Inhibitor (AZD9291) of Both Sensitizing and T790M Resistance Mutations That Spares the Wild Type Form of the Receptor(2014)591 cited
• → Discovery, Synthesis, and in Vivo Activity of a New Class of Pyrazoloquinazolines as Selective Inhibitors of Aurora B Kinase(2007)273 cited
• → Structure- and Reactivity-Based Development of Covalent Inhibitors of the Activating and Gatekeeper Mutant Forms of the Epidermal Growth Factor Receptor (EGFR)(2013)258 cited
• → SAR and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors(2005)125 cited
• → Novel inhibitors of prolyl 4-hydroxylase. 3. Inhibition by the substrate analog N-oxaloglycine and its derivatives(1992)94 cited
• → Discovery of Novel and Potent Thiazoloquinazolines as Selective Aurora A and B Kinase Inhibitors(2006)92 cited
• → A NEW CHEMICAL STRUCTURE FOR COAL(1962)47 cited
• → Synthesis and SAR of 1-acetanilide-4-aminopyrazole-substituted quinazolines: Selective inhibitors of Aurora B kinase with potent anti-tumor activity(2008)34 cited
• → Approaches to the design of anti-fibrotic drugs(1991)21 cited
• → Reaction Workup Planning: A Structured Flowchart Approach, Exemplified in Difficult Aqueous Workup of Hydrophilic Products(2014)12 cited