David J. Fairfax
Albany Molecular Research (United States)(US)
Publications by Year
Research Areas
Cyclopropane Reaction Mechanisms, Quinazolinone synthesis and applications, Catalytic Alkyne Reactions, Microwave-Assisted Synthesis and Applications, Catalytic C–H Functionalization Methods
Most-Cited Works
- → A comparative study of the decomposition of o-alkynyl-substituted aryl diazo ketones. Synthesis of polysubstituted .beta.-naphthols via arylketene intermediates(1993)56 cited
- → Scope of the Intramolecular Imidotitanium−Alkyne [2 + 2] Cycloaddition−Azatitanetine Acylation Sequence. An Efficient Procedure for the Synthesis of 2-(2-Keto-1-alkylidene)tetrahydropyrroles and Related Compounds(1997)53 cited
- → A Novel Highly Stereoselective Synthesis of 2,3-Disubstituted 3H-Quinazoline-4-one Derivatives(2007)52 cited
- → Stereo and electronic effects in the rhodium(II)-mediated synthesis of polycyclic lactones and lactams from .alpha.-diazo ester and amide precursors(1993)44 cited
- → Discovery and Preclinical Evaluation of [4-[[1-(3-fluorophenyl)methyl]-1H-indazol-5-ylamino]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamic Acid, (3S)-3-Morpholinylmethyl Ester (BMS-599626), a Selective and Orally Efficacious Inhibitor of Human Epidermal Growth Factor Receptor 1 and 2 Kinases(2009)30 cited
- → Alternatives to α-diazo ketones for tandem cyclization–cycloaddition and carbenoid–alkyne metathesis strategies. Novel cyclic enol–ether formation via carbonyl ylide rearrangement reactions(1992)30 cited
- → A General Procedure for the Synthesis of 2-Substituted Pyrimidine-5-Carboxylic Esters(2002)27 cited
- → An efficient one-pot, two-step synthesis of 4-substituted 1-heteroarylpiperazines under microwave irradiation conditions(2007)27 cited
- → An enantioselective synthesis of nitrogen protected 3-arylserine esters(2004)21 cited
- → Preparation of 5-(2-Methoxy-4-nitrophenyl)oxazole: A Key Intermediate for the Construction of VX-497(2002)21 cited