Simon Gaines
Molecular Discovery (United Kingdom)(GB)
Publications by Year
Research Areas
Magnetism in coordination complexes, Catalytic Alkyne Reactions, Nonlinear Optical Materials Research, Cyclopropane Reaction Mechanisms, Peptidase Inhibition and Analysis
Most-Cited Works
- → Large Molecular Quadratic Hyperpolarizabilities in Donor/Acceptor-Substituted trans-Tetraammineruthenium(II) Complexes(1997)68 cited
- → Identification of C-2 Hydroxyethyl Imidazopyrrolopyridines as Potent JAK1 Inhibitors with Favorable Physicochemical Properties and High Selectivity over JAK2(2013)62 cited
- → A reversed sulfonamide series of selective RORc inverse agonists(2014)35 cited
- → Identification of a sulfonamide series of CCR2 antagonists(2010)35 cited
- → Palladium-Catalyzed Ring Expansion of Spirocyclopropanes to Form Caprolactams and Azepanes(2015)24 cited
- → Irreversible 4-Aminopiperidine Transglutaminase 2 Inhibitors for Huntington's Disease(2012)20 cited
- → From PIM1 to PI3Kδ via GSK3β: Target Hopping through the Kinome(2017)16 cited
- → The identification of β-hydroxy carboxylic acids as selective MMP-12 inhibitors(2009)16 cited
- → Dopamine D3 receptor antagonists: The quest for a potentially selective PET ligand. Part one: Lead identification(2009)11 cited
- → The characterization of a novel V1b antagonist lead series(2010)4 cited