Raj Betageri
Boehringer Ingelheim (United States)(US)
Publications by Year
Research Areas
Estrogen and related hormone effects, Protein Kinase Regulation and GTPase Signaling, Inflammatory mediators and NSAID effects, Chemical Synthesis and Analysis, Enzyme Structure and Function
Most-Cited Works
- → Neutrophil rolling altered by inhibition of L-selectin shedding in vitro(1996)278 cited
- → Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand(2005)106 cited
- → Crystal Structures of the Human p56lckSH2 Domain in Complex with Two Short Phosphotyrosyl Peptides at 1.0 Å and 1.8 Å Resolution(1996)103 cited
- → Determination of Receptor-Ligand Kinetic and Equilibrium Binding Constants using Surface Plasmon Resonance: Application to the lck SH2 Domain and Phosphotyrosyl Peptides(1995)68 cited
- → Ligands for the Tyrosine Kinase p56lck SH2 Domain: Discovery of Potent Dipeptide Derivatives with Monocharged, Nonhydrolyzable Phosphate Replacements(1999)57 cited
- → Carboxymethyl-phenylalanine as a Replacement for Phosphotyrosine in SH2 Domain Binding(1998)41 cited
- → Substituted pyrazoles as novel sEH antagonist: Investigation of key binding interactions within the catalytic domain(2010)41 cited
- → Identification of Highly Efficacious Glucocorticoid Receptor Agonists with a Potential for Reduced Clinical Bone Side Effects(2014)31 cited
- → Practical synthesis of 1,3-diaryl-5-alkylpyrazoles by a highly regioselective N-arylation of 3,5-disubstituted pyrazoles with 4-fluoronitrobenzene(2000)31 cited
- → Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores(2011)19 cited