François D’Hooge
University of Oxford(GB)
Publications by Year
Research Areas
Synthesis and pharmacology of benzodiazepine derivatives, Cancer therapeutics and mechanisms, Protein Degradation and Inhibitors, HER2/EGFR in Cancer Research, Fluorine in Organic Chemistry
Most-Cited Works
- → Uptake of unnatural trehalose analogs as a reporter for Mycobacterium tuberculosis(2011)238 cited
- → ADCT-402, a PBD dimer–containing antibody drug conjugate targeting CD19-expressing malignancies(2018)175 cited
- → Genetically Encoded Azide Containing Amino Acid in Mammalian Cells Enables Site-Specific Antibody–Drug Conjugates Using Click Cycloaddition Chemistry(2015)138 cited
- → ADCT-301, a Pyrrolobenzodiazepine (PBD) Dimer–Containing Antibody–Drug Conjugate (ADC) Targeting CD25-Expressing Hematological Malignancies(2016)125 cited
- → Dye displacement assay for saccharide detection with boronate hydrogels(2008)86 cited
- → TR1801‐ADC: a highly potent cMet antibody–drug conjugate with high activity in patient‐derived xenograft models of solid tumors(2019)66 cited
- → The Development of Boronic Acids as Sensors and Separation Tools(2012)64 cited
- → Fluoroglycoproteins: ready chemical site-selective incorporation of fluorosugars into proteins(2010)52 cited
- → Antitumor Activity of MEDI3726 (ADCT-401), a Pyrrolobenzodiazepine Antibody–Drug Conjugate Targeting PSMA, in Preclinical Models of Prostate Cancer(2018)47 cited
- → Preclinical Evaluation of MEDI0641, a Pyrrolobenzodiazepine-Conjugated Antibody–Drug Conjugate Targeting 5T4(2017)45 cited