Masaki Daini
Takeda (Japan)(JP)
Publications by Year
Research Areas
Organoboron and organosilicon chemistry, Catalytic Cross-Coupling Reactions, Boron Compounds in Chemistry, Epigenetics and DNA Methylation, Crystallization and Solubility Studies
Most-Cited Works
- → Palladium-Catalyzed trans- and cis-Carboboration of Alkynes Tethered to Chloroborane with Organozirconium Reagents: Ligand-Dependent Complementary Stereoselectivity(2008)117 cited
- → Palladium-catalyzed carboboration of alkynes using chloroborane and organozirconium reagents(2008)104 cited
- → Palladium-Catalyzed, Stereoselective, Cyclizative Alkenylboration of Carbon−Carbon Double Bonds through Activation of a Boron−Chlorine Bond(2011)65 cited
- → Inhibition of KDM1A activity restores adult neurogenesis and improves hippocampal memory in a mouse model of Kabuki syndrome(2021)43 cited
- → Ruthenium-Catalyzed Dienyne Formation from Propargylic Alcohols and 1,3-Conjugated Dienes(2008)41 cited
- → LSD1 enzyme inhibitor TAK-418 unlocks aberrant epigenetic machinery and improves autism symptoms in neurodevelopmental disorder models(2021)37 cited
- → Nickel‐Catalyzed Cyclizative trans‐Carboboration of Alkynes through Activation of Boron–Chlorine Bonds by Using Organometallic Reagents as Donors of Organic Groups(2013)31 cited
- → Palladium-catalyzed Carboboration: Borylative Coupling of Alkynes with Alkenes through Activation of Boron–Chlorine Bonds(2013)23 cited
- → Design, synthesis, and structure–activity relationship of TAK-418 and its derivatives as a novel series of LSD1 inhibitors with lowered risk of hematological side effects(2022)18 cited
- → Discovery of Brain-Penetrant Glucosylceramide Synthase Inhibitors with a Novel Pharmacophore(2022)13 cited