Jean Lacrampe
Janssen (France)(FR)
Publications by Year
Research Areas
Respiratory viral infections research, Synthesis and Catalytic Reactions, Asymmetric Synthesis and Catalysis, Asthma and respiratory diseases, Fluorine in Organic Chemistry
Most-Cited Works
- → Substituted benzimidazoles with nanomolar activity against respiratory syncytial virus(2003)115 cited
- → Selection of a Respiratory Syncytial Virus Fusion Inhibitor Clinical Candidate, Part 1: Improving the Pharmacokinetic Profile Using the Structure−Property Relationship(2007)51 cited
- → Identification of R146225 as a Novel, Orally Active Inhibitor of Interleukin-5 Biosynthesis(2000)22 cited
- → Synthesis and Biological Evaluation of 1,2,4-Triazinylphenylalkylthiazolecarboxylic Acid Esters as Cytokine-Inhibiting Antedrugs with Strong Bronchodilating Effects in an Animal Model of Asthma(2004)19 cited
- JNJ-26854165 - a novel hdm2 antagonist in clinical development showing broad-spectrum preclinical antitumor activity against solid malignancies(2008)
- → Synthesis of bridged azabicyclic ketones. Solvolysis of enol ether ethylene ketal N-cholramines in acidic medium(1976)12 cited
- → Cyclisation de n-chloramines en presence d'oxyde d'argent. Synthese de molecules azapolycycliques pontees.(1975)9 cited
- → Abstract 4748: Discovery of JNJ-42756493, a potent fibroblast growth factor receptor (FGFR) inhibitor using a fragment based approach(2014)9 cited
- → Abstract 1361: Fragment based drug discovery of selective inhibitors of Fibroblast Growth Factor Receptor (FGFR)(2011)2 cited
- R170591, a New Antiviral with picoMolar Activity against Respiratory Syncytial Virus.(2001)