Goss S. Kauffman
Forma Therapeutics (United States)(US)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Synthesis and Catalytic Reactions, Synthesis and Biological Evaluation, Asymmetric Synthesis and Catalysis, HIV/AIDS drug development and treatment
Most-Cited Works
- → An Efficient Chiral Moderator Prepared from Inexpensive (+)-3-Carene: Synthesis of the HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor DPC 963(2000)193 cited
- → Rearrangement of Nα-Protected l-Asparagines with Iodosobenzene Diacetate. A Practical Route to β-Amino-l-alanine Derivatives(1997)99 cited
- → Synthesis and structure based optimization of novel Akt inhibitors(2008)75 cited
- → Synthesis of Thrombin Inhibitor DuP 714(1995)75 cited
- → Discovery and Optimization of Quinolinone Derivatives as Potent, Selective, and Orally Bioavailable Mutant Isocitrate Dehydrogenase 1 (mIDH1) Inhibitors(2019)47 cited
- → NMR Spectroscopic Investigations of Mixed Aggregates Underlying Highly Enantioselective 1,2-Additions of Lithium Cyclopropylacetylide to Quinazolinones(2001)43 cited
- → Interaction of thiamin diphosphate and thiamin thiazolone diphosphate with wheat germ pyruvate decarboxylase.(1984)38 cited
- → The discovery of highly selective erbB2 (Her2) inhibitors for the treatment of cancer(2007)25 cited
- → The chiral specific synthesis of DMP 754, a platelet GP antagonist(1996)21 cited
- → Discovery and optimization of novel piperazines as potent inhibitors of fatty acid synthase (FASN)(2019)19 cited