Ellen M. Leahy
Publications by Year
Research Areas
Blood Coagulation and Thrombosis Mechanisms, Coagulation, Bradykinin, Polyphosphates, and Angioedema, Chemical Synthesis and Analysis, Peptidase Inhibition and Analysis, Neuroendocrine Tumor Research Advances
Most-Cited Works
- → Structural Snapshots of Human HDAC8 Provide Insights into the Class I Histone Deacetylases(2004)691 cited
- → De novo design and synthesis of somatostatin non-peptide peptidomimetics utilizing .beta.-D-glucose as a novel scaffolding(1993)272 cited
- → Nonpeptidal peptidomimetics with .beta.-D-glucose scaffolding. A partial somatostatin agonist bearing a close structural relationship to a potent, selective substance P antagonist(1992)222 cited
- → Optimization of a screening lead for factor VIIa/TF(2001)45 cited
- → Potent 4-amino-5-azaindole factor VIIa inhibitors(2006)34 cited
- → Factor VIIa inhibitors: Chemical optimization, preclinical pharmacokinetics, pharmacodynamics, and efficacy in an arterial baboon thrombosis model(2006)30 cited
- → Novel 5-azaindole factor VIIa inhibitors(2006)27 cited
- → Factor VIIa inhibitors: Improved pharmacokinetic parameters(2006)13 cited
- → Efforts toward oral bioavailability in factor VIIa inhibitors(2006)9 cited
- → Crystal Structure of Human HDAC8 complexed with MS-344(2004)1 cited