Frederik Rombouts
Janssen (Belgium)(BE)
Publications by Year
Research Areas
Alzheimer's disease research and treatments, Computational Drug Discovery Methods, Catalytic Cross-Coupling Reactions, Fluorine in Organic Chemistry, Cholinesterase and Neurodegenerative Diseases
Most-Cited Works
- → In Vivo Inhibition of RIPK2 Kinase Alleviates Inflammatory Disease(2014)114 cited
- → Complementary Regioselectivity in Rh(III)-Catalyzed Insertions of Potassium Vinyltrifluoroborate via C–H Activation: Preparation and Use of 4-Trifluoroboratotetrahydroisoquinolones(2013)107 cited
- → Tau Positron Emission Tomography (PET) Imaging: Past, Present, and Future(2015)106 cited
- → Copper-Mediated Radical Trifluoromethylation of Unsaturated Potassium Organotrifluoroborates(2013)96 cited
- → Synthesis and Minisci Reactions of Organotrifluoroborato Building Blocks(2013)89 cited
- → Benzazaborinines as Novel Bioisosteric Replacements of Naphthalene: Propranolol as an Example(2015)87 cited
- → Preclinical Evaluation of18F-JNJ64349311, a Novel PET Tracer for Tau Imaging(2017)86 cited
- → 1,4-Oxazine β-Secretase 1 (BACE1) Inhibitors: From Hit Generation to Orally Bioavailable Brain Penetrant Leads(2015)77 cited
- → New evolutions in the BACE1 inhibitor field from 2014 to 2018(2019)71 cited
- → Pyrido[4,3-e][1,2,4]triazolo[4,3-a]pyrazines as Selective, Brain Penetrant Phosphodiesterase 2 (PDE2) Inhibitors(2015)56 cited