Jean‐Robert Labrosse

Publications by Year

Research Areas

Asymmetric Synthesis and Catalysis, Catalytic C–H Functionalization Methods, Catalytic Alkyne Reactions, Catalytic Cross-Coupling Reactions, Synthetic Organic Chemistry Methods

Most-Cited Works

• → Discovery of (2S)-8-[(3R)-3-Methylmorpholin-4-yl]-1-(3-methyl-2-oxobutyl)-2-(trifluoromethyl)-3,4-dihydro-2H-pyrimido[1,2-a]pyrimidin-6-one: A Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid Tumors(2014)90 cited
• → Chiral Aromatase and Dual Aromatase−Steroid Sulfatase Inhibitors from the Letrozole Template: Synthesis, Absolute Configuration, and In Vitro Activity(2008)85 cited
• → A Simple and Efficient Enantioselective Synthesis of 2-Alkylidene-3-alkyl-1,4-benzodioxanes by Palladium-Catalyzed Annulation of Benzene-1,2-diol and Propargylic Carbonates(2000)65 cited
• → An easy palladium-catalyzed access to 2-alkylidene-1,4-benzodioxanes(1999)64 cited
• → Palladium-Catalyzed Synthesis of 2,3-Dihydro-2-ylidene-1,4-benzodioxins(2001)53 cited
• → Asymmetric palladium(0)-mediated synthesis of 2-vinylchroman(1999)43 cited
• → Pd-Catalyzed annulation of benzene-1,2-diol and propargylic carbonates: a new example of asymmetric catalysis(2003)37 cited
• → Bicyclic Derivatives of the Potent Dual Aromatase–Steroid Sulfatase Inhibitor 2‐Bromo‐4‐{[(4‐cyanophenyl)(4H‐1,2,4‐triazol‐4‐yl)amino]methyl}phenylsulfamate: Synthesis, SAR, Crystal Structure, and in vitro and in vivo Activities(2010)25 cited
• → Palladium‐Catalyzed Annulation of Aryl‐1,2‐diols and Propargylic Carbonates. Theoretical Study of the Observed Regioselectivities(2003)23 cited
• → Asymmetric palladium-catalyzed annulation of benzene-1,2-diol and racemic secondary propargylic carbonates bearing two different substituents(2005)22 cited