Younes Bekkali
Boehringer Ingelheim (United States)(US)
Publications by Year
Research Areas
Estrogen and related hormone effects, Protease and Inhibitor Mechanisms, Inflammatory mediators and NSAID effects, Hormonal Regulation and Hypertension, Peptidase Inhibition and Analysis
Most-Cited Works
- → Design and Synthesis of Dipeptide Nitriles as Reversible and Potent Cathepsin S Inhibitors(2002)83 cited
- → Discovery and SAR study of novel dihydroquinoline-containing glucocorticoid receptor agonists(2007)48 cited
- → Quinol-4-ones as Steroid A-Ring Mimetics in Nonsteroidal Dissociated Glucocorticoid Agonists(2006)41 cited
- → Discovery and SAR study of novel dihydroquinoline containing glucocorticoid receptor ligands(2005)35 cited
- → Identification of dissociated non-steroidal glucocorticoid receptor agonists(2007)34 cited
- → Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores(2011)19 cited
- → Identification of a novel class of succinyl-nitrile-based Cathepsin S inhibitors(2007)12 cited
- → Theoretical and experimental approaches to the effects of solvation on the small internal rotational potential of benzal fluoride(1996)6 cited
- → Design and Synthesis of Dipeptide Nitriles as Reversible and Potent Cathepsin S Inhibitors.(2003)6 cited
- → Cathepsin S complexed with Compound 15(2007)