Takanori Koike
Astellas Pharma (Japan)(JP)
Publications by Year
Research Areas
Legal and Regulatory Analysis, Linguistic, Cultural, and Literary Studies, Military Technology and Strategies, Catalytic Cross-Coupling Reactions, Chemical synthesis and alkaloids
Most-Cited Works
- → Lipase-catalyzed preparation of both enantiomers of methyl jasmonate(2001)43 cited
- → Design, synthesis and biological activity of selective and orally available TF/FVIIa complex inhibitors containing non-amidine P1 ligands(2006)20 cited
- → Syntheses and odour descriptions of jasmine lactone and cis‐jasmone analogues bearing cyclopropane moieties(2001)20 cited
- → One‐Pot Preparation of Unsymmetrical Biaryls via Suzuki Cross‐Coupling Reaction of Aryl Halide using Phase‐Transfer Catalyst in a Biphasic Solvent System(2007)16 cited
- → One‐Pot Synthetic Procedure for2,2′‐Disubstituted Biaryls via the Suzuki Coupling Reaction of Aryl Triflates in a Biphasic Solvent System(2006)15 cited
- → Potent and selective TF/FVIIa inhibitors containing a neutral P1 ligand(2006)15 cited
- → Discovery and biological evaluation of 1-{2,7-diazaspiro[3.5]nonan-2-yl}prop-2-en-1-one derivatives as covalent inhibitors of KRAS G12C with favorable metabolic stability and anti-tumor activity(2022)14 cited
- → Discovery and structure-activity relationships study of positive allosteric modulators of the M3 muscarinic acetylcholine receptor(2020)10 cited
- → Syntheses and odour descriptions of cyclopropanated compounds 2.1 Analogues of methyl jasmonate(2002)9 cited
- → Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure–activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl}prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors(2023)5 cited