Fabrizio Manetti
University of Siena(IT)
Publications by Year
Research Areas
Synthesis and biological activity, Receptor Mechanisms and Signaling, Tuberculosis Research and Epidemiology, HIV/AIDS drug development and treatment, Cancer therapeutics and mechanisms
Most-Cited Works
- → MmpL3 Is the Cellular Target of the Antitubercular Pyrrole Derivative BM212(2011)210 cited
- → Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones(2009)158 cited
- → Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis(2008)141 cited
- → Synthesis, Biological Evaluation, and Pharmacophore Generation of New Pyridazinone Derivatives with Affinity toward α1- and α2-Adrenoceptors(2001)120 cited
- → LIM kinases are attractive targets with many macromolecular partners and only a few small molecule regulators(2011)114 cited
- → Antimycobacterial Agents. Novel Diarylpyrrole Derivatives of BM212 Endowed with High Activity toward Mycobacterium tuberculosis and Low Cytotoxicity(2006)114 cited
- → Toward the Discovery of Novel Anti‐HIV Drugs. Second‐Generation Inhibitors of the Cellular ATPase DDX3 with Improved Anti‐HIV Activity: Synthesis, Structure–Activity Relationship Analysis, Cytotoxicity Studies, and Target Validation(2011)105 cited
- → 4-Hydroxyphenylpyruvate Dioxygenase and Its Inhibition in Plants and Animals: Small Molecules as Herbicides and Agents for the Treatment of Human Inherited Diseases(2017)104 cited
- → Improved BM212 MmpL3 Inhibitor Analogue Shows Efficacy in Acute Murine Model of Tuberculosis Infection(2013)94 cited
- → Acylthiourea, Acylurea, and Acylguanidine Derivatives with Potent Hedgehog Inhibiting Activity(2012)88 cited