Elisabeth Klaasse
Leiden University(NL)Centre for Human Drug Research(NL)
Publications by Year
Research Areas
Receptor Mechanisms and Signaling, Cardiac electrophysiology and arrhythmias, Adenosine and Purinergic Signaling, Ion channel regulation and function, Neuropeptides and Animal Physiology
Most-Cited Works
- → Internalization and desensitization of adenosine receptors(2007)120 cited
- → Prospective Validation of a Comprehensive In silico hERG Model and its Applications to Commercial Compound and Drug Databases(2010)108 cited
- → N6-Cyclopentyl-2-(3-phenylaminocarbonyltriazene-1-yl)adenosine (TCPA), a Very Selective Agonist with High Affinity for the Human Adenosine A1 Receptor(2003)45 cited
- → Strategies To Reduce hERG K+ Channel Blockade. Exploring Heteroaromaticity and Rigidity in Novel Pyridine Analogues of Dofetilide(2013)37 cited
- → Removal of Human Ether-à-go-go Related Gene (hERG) K+ Channel Affinity through Rigidity: A Case of Clofilium Analogues(2013)32 cited
- → Exploring Chemical Substructures Essential for hERG K+ Channel Blockade by Synthesis and Biological Evaluation of Dofetilide Analogues(2009)26 cited
- → Allosteric modulators of the hERG K+ channel(2013)23 cited
- → Allosteric modulators affect the internalization of human adenosine A1 receptors(2005)20 cited
- → Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E‐4031 Analogues(2011)19 cited
- → Characterization of [3H]LUF5834: A novel non-ribose high-affinity agonist radioligand for the adenosine A1 receptor(2010)13 cited