Nicolas Proisy
Publications by Year
Research Areas
Computational Drug Discovery Methods, Heat shock proteins research, DNA Repair Mechanisms, Protein Kinase Regulation and GTPase Signaling, Lung Cancer Treatments and Mutations
Most-Cited Works
- → Inhibition of Hsp90 with Synthetic Macrolactones: Synthesis and Structural and Biological Evaluation of Ring and Conformational Analogs of Radicicol(2006)66 cited
- → Structure-Guided Evolution of Potent and Selective CHK1 Inhibitors through Scaffold Morphing(2011)59 cited
- → Multiparameter Lead Optimization to Give an Oral Checkpoint Kinase 1 (CHK1) Inhibitor Clinical Candidate: (R)-5-((4-((Morpholin-2-ylmethyl)amino)-5-(trifluoromethyl)pyridin-2-yl)amino)pyrazine-2-carbonitrile (CCT245737)(2016)37 cited
- → Synthetic ansamycins prepared by a ring-expanding Claisen rearrangement. Synthesis and biological evaluation of ring and conformational analogues of the Hsp90 molecular chaperone inhibitor geldanamycin(2007)21 cited
- → Multi-parameter lead optimization to give an oral CHK1 inhibitor clinical candidate: (R)-5-((4-((morpholin-2-ylmethyl)amino)-5-(trifluoromethyl)pyridin-2-yl)amino)pyrazine-2-carbonitrile (CCT245737)(2015)
- → CCDC 624769: Experimental Crystal Structure Determination(2007)