Didier Berthelot
Janssen (Belgium)(BE)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Catalytic C–H Functionalization Methods, Computational Drug Discovery Methods, Catalytic Cross-Coupling Reactions, Radical Photochemical Reactions
Most-Cited Works
- → γ-Secretase Modulators as Potential Disease Modifying Anti-Alzheimer’s Drugs(2010)160 cited
- → 2-Amino-3,4-dihydroquinazolines as Inhibitors of BACE-1 (β-Site APP Cleaving Enzyme): Use of Structure Based Design to Convert a Micromolar Hit into a Nanomolar Lead(2007)145 cited
- → Analogues of Morphanthridine and the Tear Gas Dibenz[b,f][1,4]oxazepine (CR) as Extremely Potent Activators of the Human Transient Receptor Potential Ankyrin 1 (TRPA1) Channel(2010)94 cited
- → The accelerated development of an optimized synthesis of 1,2,4-oxadiazoles: application of microwave irradiation and statistical design of experiments(2003)77 cited
- → Minisci-Photoredox-Mediated α-Heteroarylation of N-Protected Secondary Amines: Remarkable Selectivity of Azetidines(2018)74 cited
- → Design and Synthesis of a Novel Series of Bicyclic Heterocycles As Potent γ-Secretase Modulators(2012)60 cited
- → Ruthenium‐Catalyzed α‐(Hetero)Arylation of Saturated Cyclic Amines: Reaction Scope and Mechanism(2013)60 cited
- → Tricyclic 3,4-dihydropyrimidine-2-thione derivatives as potent TRPA1 antagonists(2011)58 cited
- → Removal of the Pyridine Directing Group from α-Substituted N-(Pyridin-2-yl)piperidines Obtained via Directed Ru-Catalyzed sp3 C–H Functionalization(2013)57 cited
- → Iron-Catalyzed Synthesis of Sulfur-Containing Heterocycles(2016)25 cited