Steven M. Bromidge
Evotec (United Kingdom)(GB)
Publications by Year
Research Areas
Receptor Mechanisms and Signaling, Synthesis and Biological Evaluation, Neurotransmitter Receptor Influence on Behavior, Phenothiazines and Benzothiazines Synthesis and Activities, Pharmacological Receptor Mechanisms and Effects
Most-Cited Works
- → SB 242084, a Selective and Brain Penetrant 5-HT 2C Receptor Antagonist(1997)523 cited
- → Characterization of SB‐269970‐A, a selective 5‐HT7 receptor antagonist(2000)283 cited
- → A Novel, Potent, and Selective 5-HT7Antagonist: (R)-3-(2-(2-(4-Methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulfonyl)phenol (SB-269970)(2000)249 cited
- → SB-399885 is a potent, selective 5-HT6 receptor antagonist with cognitive enhancing properties in aged rat water maze and novel object recognition models(2006)229 cited
- → Binding Mode and Structure–Activity Relationships around Direct Inhibitors of the Nrf2–Keap1 Complex(2014)170 cited
- → 5-Chloro-N-(4-methoxy-3-piperazin-1-yl- phenyl)-3-methyl-2-benzothiophenesulfon- amide (SB-271046): A Potent, Selective, and Orally Bioavailable 5-HT6 Receptor Antagonist(1999)170 cited
- → Characterization of SB‐271046: A potent, selective and orally active 5‐HT6 receptor antagonist(2000)136 cited
- → Characterization of [125I]‐SB‐258585 binding to human recombinant and native 5‐HT6 receptors in rat, pig and human brain tissue(2000)120 cited
- → SB-243213; a selective 5-HT2C receptor inverse agonist with improved anxiolytic profile: lack of tolerance and withdrawal anxiety(2001)100 cited
- → 6-Chloro-5-methyl-1-[[2-[(2-methyl-3- pyridyl)oxy]-5-pyridyl]carbamoyl]indoline (SB-242084): The First Selective and Brain Penetrant 5-HT2C Receptor Antagonist(1997)84 cited