Helen J. Mason
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Blood Coagulation and Thrombosis Mechanisms, Phosphodiesterase function and regulation, Asymmetric Synthesis and Catalysis, Chemical Synthesis and Reactions
Most-Cited Works
- → Parallel Synthesis of Aldehydes and Ketone Facilitated by a New Solid-Phase Weinreb Amide(1999)49 cited
- → Substituted Pyrazolopyridines as Potent and Selective PDE5 Inhibitors: Potential Agents for Treatment of Erectile Dysfunction(2001)45 cited
- → Design and Structure−Activity Relationships of Potent and Selective Inhibitors of Blood Coagulation Factor Xa(1999)42 cited
- → An Imidazopiperidine Series of CCR5 Antagonists for the Treatment of HIV: The Discovery of N-{(1S)-1-(3-Fluorophenyl)-3-[(3-endo)-3-(5-isobutyryl-2-methyl-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]propyl}acetamide (PF-232798)(2010)40 cited
- → Substituted Pyrazolopyridopyridazines as Orally Bioavailable Potent and Selective PDE5 Inhibitors: Potential Agents for Treatment of Erectile Dysfunction(2003)37 cited
- → Sulfonamidopyrrolidinone Factor Xa Inhibitors: Potency and Selectivity Enhancements via P-1 and P-4 Optimization(1999)36 cited
- → Optimisation of a novel series of selective CNS penetrant CB2 agonists(2011)26 cited
- → Synthesis, SAR and in vivo activity of novel thienopyridine sulfonamide pyrrolidinones as factor Xa inhibitors(1999)25 cited
- → Synthesis of fused pyridopyrrolidine dione derivatives using hetero Diels–Alder reactions(2001)24 cited
- → Aminoisoquinolines: Design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA(1999)22 cited