Nicole Blaquière
Publications by Year
Research Areas
Catalytic C–H Functionalization Methods, NF-κB Signaling Pathways, Protein Degradation and Inhibitors, Ubiquitin and proteasome pathways, Cytokine Signaling Pathways and Interactions
Most-Cited Works
- → Ruthenium-Catalyzed Dehydrogenation of Ammonia Boranes(2008)303 cited
- → Discovery of 2-{3-[2-(1-Isopropyl-3-methyl-1H-1,2–4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl]-1H-pyrazol-1-yl}-2-methylpropanamide (GDC-0032): A β-Sparing Phosphoinositide 3-Kinase Inhibitor with High Unbound Exposure and Robust in Vivo Antitumor Activity(2013)175 cited
- → Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1: Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties(2021)144 cited
- → NF-κB inducing kinase is a therapeutic target for systemic lupus erythematosus(2018)125 cited
- → Rapid Synthesis of 1,3,5-Substituted 1,2,4-Triazoles from Carboxylic Acids, Amidines, and Hydrazines(2011)109 cited
- → Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα)(2019)104 cited
- → Four‐Component Synthesis of Fully Substituted 1,2,4‐Triazoles(2009)97 cited
- → Decarboxylative Ketone Aldol Reactions: Development and Mechanistic Evaluation under Metal-Free Conditions(2009)80 cited
- → Direct intramolecular arylation of unactivated arenes: application to the synthesis of aporphine alkaloids(2004)73 cited
- → Monomeric Targeted Protein Degraders(2020)62 cited