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Gary L. Grunewald | doi.page

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Gary L. Grunewald

University of Kansas(US)

Publications by Year

Research Areas

Synthesis and Biological Activity, Chemical Synthesis and Analysis, Berberine and alkaloids research, Chemical synthesis and alkaloids, Carbohydrate Chemistry and Synthesis

Most-Cited Works

→ The Chemistry of Barrelene. III. A Unique Photoisomerization to Semibullvalene(1966)213 cited
→ "Hydrophobic collapse" of taxol and Taxotere solution conformations in mixtures of water and organic solvent(1993)149 cited
→ Mechanistic and exploratory organic photochemistry. XLIV. The barrelene to semibullvalene transformation. Correlation of excited-state potential energy surfaces with reactivity(1969)94 cited
→ Synthesis and physical properties of barrelene, a unique Moebius-like molecule(1969)80 cited
→ Effect of Ring Size or an Additional Heteroatom on the Potency and Selectivity of Bicyclic Benzylamine-Type Inhibitors of PhenylethanolamineN-Methyltransferase1a(1996)76 cited
→ Getting the Adrenaline Going(2001)59 cited

→ Application of the Goldilocks Effect to the Design of Potent and Selective Inhibitors of PhenylethanolamineN-Methyltransferase: Balancing pK_aand Steric Effects in the Optimization of 3-Methyl-1,2,3,4-tetrahydroisoquinoline Inhibitors by β-Fluorination(2006)

51 cited

→ Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors(2010)45 cited

→ Synthesis and Biochemical Evaluation of 3-Fluoromethyl-1,2,3,4-tetrahydroisoquinolines as Selective Inhibitors of Phenylethanolamine N-Methyltransferase versus the α₂-Adrenoceptor(1999)44 cited

→ The NH---FC Dipole Orientation Effect for Pendant Exocyclic CH₂F(2002)42 cited