Jeffrey Y. Melamed
United States Military Academy(US)
Publications by Year
Research Areas
HIV Research and Treatment, HIV/AIDS drug development and treatment, Biochemical and Molecular Research, Asymmetric Synthesis and Catalysis, HIV/AIDS Research and Interventions
Most-Cited Works
- → Diketo acid inhibitor mechanism and HIV-1 integrase: Implications for metal binding in the active site of phosphotransferase enzymes(2002)395 cited
- → HIV-1 integrase inhibitors that compete with the target DNA substrate define a unique strand transfer conformation for integrase(2000)317 cited
- → 4-Aryl-2,4-dioxobutanoic Acid Inhibitors of HIV-1 Integrase and Viral Replication in Cells(2000)187 cited
- → Synthesis and Evaluation of Heterocyclic Catechol Mimics as Inhibitors of Catechol-O-methyltransferase (COMT)(2015)45 cited
- → A potent and orally active HIV-1 integrase inhibitor(2006)36 cited
- → Total Synthesis of (−)-Normalindine via Addition of Metalated 4-Methyl-3-cyanopyridine to an Enantiopure Sulfinimine(2006)33 cited
- → Synthesis and evaluation of a new series of Neuropeptide S receptor antagonists(2010)26 cited
- → Synthesis of 5-(1-H or 1-alkyl-5-oxopyrrolidin-3-yl)-8-hydroxy-[1,6]-naphthyridine-7-carboxamide inhibitors of HIV-1 integrase(2008)24 cited
- → Total Synthesis of (‐)‐Normalindine via Addition of Metalated 4‐Methyl‐3‐cyanopyridine to an Enantiopure Sulfinimine.(2007)