Iolanda Micco
Publications by Year
Research Areas
Nicotinic Acetylcholine Receptors Study, Receptor Mechanisms and Signaling, Chemical Synthesis and Analysis, Cholinesterase and Neurodegenerative Diseases, Synthesis and Biological Evaluation
Most-Cited Works
- → Screening of DNA-Encoded Small Molecule Libraries inside a Living Cell(2021)80 cited
- → An overview of DNA-encoded libraries: A versatile tool for drug discovery(2020)73 cited
- → SAR and biological evaluation of SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist(2009)41 cited
- → Novel Alpha-7 Nicotinic Acetylcholine Receptor Agonists Containing a Urea Moiety: Identification and Characterization of the Potent, Selective, and Orally Efficacious Agonist 1-[6-(4-Fluorophenyl)pyridin-3-yl]-3-(4-piperidin-1-ylbutyl) Urea (SEN34625/WYE-103914)(2010)30 cited
- → Discovery of a Novel Alpha-7 Nicotinic Acetylcholine Receptor Agonist Series and Characterization of the Potent, Selective, and Orally Efficacious Agonist 5-(4-Acetyl[1,4]diazepan-1-yl)pentanoic Acid [5-(4-Methoxyphenyl)-1H-pyrazol-3-yl] Amide (SEN15924, WAY-361789)(2012)26 cited
- → 2,9-Disubstituted-N6-(arylcarbamoyl)-8-azaadenines as new selective A3 adenosine receptor antagonists: Synthesis, biochemical and molecular modelling studies(2005)21 cited
- → Design and synthesis of a hybrid series of potent and selective agonists of α7 nicotinic acetylcholine receptor(2014)21 cited
- → N-[5-(5-Fluoropyridin-3-yl)-1H-pyrazol-3-yl]-4-piperidin-1-ylbutyramide (SEN78702, WYE-308775): A Medicinal Chemistry Effort toward an α7 Nicotinic Acetylcholine Receptor Agonist Preclinical Candidate(2012)14 cited
- → Searching for Dual Inhibitors of the MDM2‐p53 and MDMX‐p53 Protein–Protein Interaction by a Scaffold‐Hopping Approach(2014)13 cited
- → A Homogeneous HTRF Assay for the Identification of Inhibitors of the TWEAK-Fn14 Protein Interaction(2012)11 cited