Akiyasu Kouketsu
Publications by Year
Research Areas
Histone Deacetylase Inhibitors Research, Protein Degradation and Inhibitors, Peptidase Inhibition and Analysis, Click Chemistry and Applications, Chemical Synthesis and Analysis
Most-Cited Works
- → Novel Inhibitors of Human Histone Deacetylases: Design, Synthesis, Enzyme Inhibition, and Cancer Cell Growth Inhibition of SAHA-Based Non-hydroxamates(2005)109 cited
- → Highly Potent and Selective Histone Deacetylase 6 Inhibitors Designed Based on a Small-Molecular Substrate(2006)104 cited
- → Design, Synthesis, Structure−Selectivity Relationship, and Effect on Human Cancer Cells of a Novel Series of Histone Deacetylase 6-Selective Inhibitors(2007)102 cited
- → Thiol-based SAHA analogues as potent histone deacetylase inhibitors(2004)92 cited
- → Identification of a potent non-hydroxamate histone deacetylase inhibitor by mechanism-based drug design(2004)61 cited
- → Design and synthesis of non-hydroxamate histone deacetylase inhibitors: identification of a selective histone acetylating agent(2005)26 cited
- → A Practical Synthesis of (S)-tert-Butyl 3-Methyl-1,4-diazepane-1-carboxylate, the Key Intermediate of Rho–Kinase Inhibitor K-115(2012)12 cited
- → Thiol‐Based SAHA Analogues as Potent Histone Deacetylase Inhibitors.(2004)1 cited
- P-440 DISCOVERY OF NOVEL HISTONE DEACETYLASE 6 SELECTIVE INHIBITORS(2006)