Martin Duplessis
Aegera Therapeutics (Canada)(CA)
Publications by Year
Research Areas
Cyclopropane Reaction Mechanisms, HIV/AIDS drug development and treatment, Catalytic Cross-Coupling Reactions, Catalytic C–H Functionalization Methods, HIV Research and Treatment
Most-Cited Works
- → Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide (CPI-1205), a Potent and Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymphomas(2016)218 cited
- → Identification of a genetic determinant responsible for host specificity in Streptococcus thermophilus bacteriophages(2001)179 cited
- → Arylcyclopropanes: Properties, Synthesis and Use in Medicinal Chemistry(2010)122 cited
- → Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains(2016)118 cited
- → Genomic Organization and Molecular Analysis of Virulent Bacteriophage 2972 Infecting an Exopolysaccharide-Producing Streptococcus thermophilus Strain(2005)87 cited
- → Direct N-Cyclopropylation of Cyclic Amides and Azoles Employing a Cyclopropylbismuth Reagent(2006)78 cited
- → Discovery, design, and synthesis of indole-based EZH2 inhibitors(2015)64 cited
- → Palladium-Catalyzed Cross-Coupling Reaction of Tricyclopropylbismuth with Aryl Halides and Triflates(2008)58 cited
- → Global gene expression analysis of two Streptococcus thermophilus bacteriophages using DNA microarray(2005)48 cited
- → Characterization of Streptococcus thermophilus Host Range Phage Mutants(2006)41 cited