Paul D. Greenspan
Tri-City Medical Center(US)
Publications by Year
Research Areas
Synthetic Organic Chemistry Methods, Protease and Inhibitor Mechanisms, Melanoma and MAPK Pathways, Traditional and Medicinal Uses of Annonaceae, Peptidase Inhibition and Analysis
Most-Cited Works
- → A small-molecule inhibitor of the ubiquitin activating enzyme for cancer treatment(2018)441 cited
- → Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer(2021)197 cited
- → Identification of Dipeptidyl Nitriles as Potent and Selective Inhibitors of Cathepsin B through Structure-Based Drug Design(2001)136 cited
- → An unusual oxidative cyclization. A synthesis and absolute stereochemical assignment of (-)-rocaglamide(1990)103 cited
- → A Total Synthesis of ( + )‐2′S, 3′R‐Zoapatanol(1994)41 cited
- → Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route(2021)41 cited
- → Diastereoselective diels-alder reactions between substituted 1,3-butadienes and n-α-methylbenzylmaleimide(1991)35 cited
- → Triphenylsilanol as a water surrogate for regioselective Pd catalyzed allylations(1993)35 cited
- → Design and Optimization of Potent and Orally Bioavailable Tetrahydronaphthalene Raf Inhibitors(2011)33 cited
- → N-Arylaminonitriles as bioavailable peptidomimetic inhibitors of cathepsin B(2003)28 cited