Allan Dishington
Jacobs (United Kingdom)(GB)
Publications by Year
Research Areas
Asymmetric Synthesis and Catalysis, Crystallization and Solubility Studies, X-ray Diffraction in Crystallography, Asymmetric Hydrogenation and Catalysis, Sulfur-Based Synthesis Techniques
Most-Cited Works
- → The Identification of Potent, Selective, and Orally Available Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase: The Discovery of AZD0156 (8-{6-[3-(Dimethylamino)propoxy]pyridin-3-yl}-3-methyl-1-(tetrahydro-2H-pyran-4-yl)-1,3-dihydro-2H-imidazo[4,5-c]quinolin-2-one)(2018)115 cited
- → Discovery of AZD4573, a Potent and Selective Inhibitor of CDK9 That Enables Short Duration of Target Engagement for the Treatment of Hematological Malignancies(2020)100 cited
- → Discovery of Novel 3-Quinoline Carboxamides as Potent, Selective, and Orally Bioavailable Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase(2016)74 cited
- → Pyrimidinone Nicotinamide Mimetics as Selective Tankyrase and Wnt Pathway Inhibitors Suitable for in Vivo Pharmacology(2015)65 cited
- → Rapid Generation of a High Quality Lead for Transforming Growth Factor-β (TGF-β) Type I Receptor (ALK5)(2009)43 cited
- → Sulfonyl-morpholino-pyrimidines: SAR and development of a novel class of selective mTOR kinase inhibitor(2012)33 cited
- → Discovery of a Series of 3-Cinnoline Carboxamides as Orally Bioavailable, Highly Potent, and Selective ATM Inhibitors(2018)29 cited
- → Neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase(2007)25 cited
- → Discovery of a Series of 7-Azaindoles as Potent and Highly Selective CDK9 Inhibitors for Transient Target Engagement(2021)24 cited
- → Synthesis of Functionalized Cyanopyrazoles via Magnesium Bases(2014)18 cited