Curt D. Haffner
RWTH Aachen University(DE)
Publications by Year
Research Areas
Estrogen and related hormone effects, Hormonal Regulation and Hypertension, Steroid Chemistry and Biochemistry, Peptidase Inhibition and Analysis, Calcium signaling and nucleotide metabolism
Most-Cited Works
- → Identification of a Chemical Tool for the Orphan Nuclear Receptor FXR(2000)521 cited
- → Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)—synthesis and biological activity(2003)311 cited
- → Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors(2015)130 cited
- → Pyrrolidinyl pyridone and pyrazinone analogues as potent inhibitors of prolyl oligopeptidase (POP)(2008)60 cited
- → 6-Azasteroids: Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase(1994)59 cited
- → Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38(2015)54 cited
- → The Palladium-Catalyzed Enyne Cycloisomerization Reaction in a General Approach to the Asymmetric Syntheses of the Picrotoxane Sesquiterpenes. Part I. First-Generation Total Synthesis of Corianin and Formal Syntheses of Picrotoxinin and Picrotin(1999)53 cited
- → 6-Azasteroids: potent dual inhibitors of human type 1 and 2 steroid 5.alpha.-reductase(1993)52 cited
- → Structure-Based Design of Potent Retinoid X Receptor α Agonists(2004)48 cited
- → Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase by 6-Azaandrost-4-en-3-ones: Optimization of the C17 Substituent(1995)47 cited