George V. Delucca
Bristol-Myers Squibb (United States)(US)
Publications by Year
Research Areas
Asthma and respiratory diseases, HIV/AIDS drug development and treatment, Multiple Myeloma Research and Treatments, Protein Degradation and Inhibitors, HIV Research and Treatment
Most-Cited Works
- → Cyclic HIV Protease Inhibitors: Synthesis, Conformational Analysis, P2/P2‘ Structure−Activity Relationship, and Molecular Recognition of Cyclic Ureas(1996)170 cited
- → CCR3 antagonists: a potential new therapy for the treatment of asthma. Discovery and structure–activity relationships(2002)46 cited
- → Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design(2021)42 cited
- → From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part I: The discovery of CCR3 antagonist development candidate BMS-639623 with picomolar inhibition potency against eosinophil chemotaxis(2007)30 cited
- → Development of BET Inhibitors as Potential Treatments for Cancer: Optimization of Pharmacokinetic Properties(2022)10 cited
- → Discovery and synthesis of cyclohexenyl derivatives as modulators of CC chemokine receptor 2 activity(2015)4 cited
- → CCDC 1419348: Experimental Crystal Structure Determination(2015)