Peter H. Dorff
Pfizer (United States)(US)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Synthesis and Biological Evaluation, Bioactive Compounds and Antitumor Agents, Drug Transport and Resistance Mechanisms, Carbohydrate Chemistry and Synthesis
Most-Cited Works
- → Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active γ-Secretase Inhibitor(2012)420 cited
- → A solid phase CBZ chloride equivalent — a new matrix specific linker(1995)113 cited
- → Metabolism-Directed Design of Oxetane-Containing Arylsulfonamide Derivatives as γ-Secretase Inhibitors(2011)105 cited
- → Mammalian topoisomerase II inhibitory activity of 1-cyclopropyl-6,8-difluoro-1,4-dihydro-7-(2,6-dimethyl-4-pyridinyl)-4-oxo-3-quinolinecarboxylic acid and related derivatives(1993)73 cited
- → Discovery and Optimization of a Novel Spiropyrrolidine Inhibitor of β-Secretase (BACE1) through Fragment-Based Drug Design(2012)63 cited
- → Deprotection of N-Boc Groups under Continuous-Flow High-Temperature Conditions(2019)47 cited
- → Preparation and reactions of chiral propargylic amines(1992)47 cited
- → 3-Quinolinecarboxamides. A series of novel orally-active antiherpetic agents(1993)35 cited
- → Synthesis and Antibacterial Activity of Some Novel 1-Substituted 1,4-Dihydro-4-oxo-7-pyridinyl-3-quinolinecarboxylic Acids. Potent Antistaphylococcal Agents(1995)31 cited
- → Novel solid-phase preparation of 2,6,9-trisubstituted purines for combinatorial library generation(2001)30 cited