Dianna Lester-Zeiner
Rapt Therapeutics (United States)(US)APT Therapeutics (United States)(US)
Publications by Year
Research Areas
Phosphodiesterase function and regulation, Coagulation, Bradykinin, Polyphosphates, and Angioedema, Cholinesterase and Neurodegenerative Diseases, Neuropeptides and Animal Physiology, Receptor Mechanisms and Signaling
Most-Cited Works
- → Identification of potent, noncovalent fatty acid amide hydrolase (FAAH) inhibitors(2011)48 cited
- → Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)(2013)43 cited
- → Discovery of Clinical Candidate 1-(4-(3-(4-(1H-Benzo[d]imidazole-2-carbonyl)phenoxy)pyrazin-2-yl)piperidin-1-yl)ethanone (AMG 579), A Potent, Selective, and Efficacious Inhibitor of Phosphodiesterase 10A (PDE10A)(2014)36 cited
- → Rapid Identification of a Novel Small Molecule Phosphodiesterase 10A (PDE10A) Tracer(2012)28 cited
- → Identification of a Nonpeptidic and Conformationally Restricted Bradykinin B1 Receptor Antagonist with Anti-Inflammatory Activity(2007)26 cited
- → Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides(2007)26 cited
- → Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)(2014)25 cited
- → Aryl sulfones as novel Bradykinin B1 receptor antagonists for treatment of chronic pain(2008)20 cited
- → AMG 580: A Novel Small Molecule Phosphodiesterase 10A (PDE10A) Positron Emission Tomography Tracer(2014)18 cited
- → A new class of bradykinin 1 receptor antagonists containing the piperidine acetic acid tetralin core(2006)18 cited