Jacques Guillaume
IAIN Palangka Raya(ID)
Publications by Year
Research Areas
Synthesis and Biological Evaluation, Chemical Reaction Mechanisms, Renin-Angiotensin System Studies, Receptor Mechanisms and Signaling, Synthesis and pharmacology of benzodiazepine derivatives
Most-Cited Works
- → Sulfonylureas and Sulfonylcarbamates as New Non-Tetrazole Angiotensin II Receptor Antagonists. Discovery of a Highly Potent Orally Active (Imidazolylbiphenylyl)sulfonylurea (HR 720)(1995)64 cited
- → (Tétrahydro-1,2,3,6 pyridinyl-4)-3 1H-indoles: synthèse, propriétés sérotoninergique et anti-dopaminergiques(1987)33 cited
- → Balanced AT1 and AT2 angiotensin II antagonists. I. New orally active 5-carboxyl imidazolyl biphenyl sulfonylureas(1995)17 cited
- → Thiol inhibitors of endothelin-converting enzyme(1996)11 cited
- → Porcine D-amino acid oxidase: Production of the biologically active enzyme in Escherichia coli(1989)10 cited
- → Balanced AT1 and AT2 angiotensin II antagonists. III. potent and orally active 5-β-ketosulfoxide imidazolyl biphenyl sulfonylureas(1995)10 cited
- → Balanced AT1 and AT2 angiotensin II antagonists. II. Potent 5 α-hydroxyacid imidazolyl biphenyl sulfonylureas(1995)8 cited
- → New Heterocycles-Acces to Thieno[3,2-b][f]- and Thieno[2,3-b][f]benzazepine Derivatives(1981)8 cited
- [Mutagenesis of the human histamine H1 receptor and design of new antihistamine agents].(1996)
- → ChemInform Abstract: Sulfonylureas and Sulfonylcarbamates as New Non‐Tetrazole Angiotensin II Receptor Antagonists. Discovery of a Highly Potent Orally Active ( Imidazolylbiphenylyl)sulfonylurea (HR 720) (II).(1995)1 cited