Xiaoyun Lu
Sun Yat-sen University(CN)Jinan University(CN)Ministry of Education(TH)Annoroad Gene Technology (China)(CN)Jinan University(LB)South China University of Technology(CN)
Publications by Year
Research Areas
Cancer therapeutics and mechanisms, Lung Cancer Treatments and Mutations, Protein Degradation and Inhibitors, Quinazolinone synthesis and applications, Computational Drug Discovery Methods
Most-Cited Works
- → Constructing a synthetic pathway for acetyl-coenzyme A from one-carbon through enzyme design(2019)267 cited
- → Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region–Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib(2013)175 cited
- → New Promise and Opportunities for Allosteric Kinase Inhibitors(2019)163 cited
- → Targeting EGFRL858R/T790M and EGFRL858R/T790M/C797S resistance mutations in NSCLC: Current developments in medicinal chemistry(2018)156 cited
- → Discovery and Optimization of 3-(2-(Pyrazolo[1,5-a]pyrimidin-6-yl)ethynyl)benzamides as Novel Selective and Orally Bioavailable Discoidin Domain Receptor 1 (DDR1) Inhibitors(2013)155 cited
- → Design, Synthesis, and in Vitro Biological Evaluation of 1H-1,2,3-Triazole-4-carboxamide Derivatives as New Anti-influenza A Agents Targeting Virus Nucleoprotein