John P. Mallamo
Publications by Year
Research Areas
Asymmetric Synthesis and Catalysis, Calpain Protease Function and Regulation, Chemical Synthesis and Analysis, Angiogenesis and VEGF in Cancer, Synthetic Organic Chemistry Methods
Most-Cited Works
- → Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery(2011)433 cited
- → Knowledge Based Prediction of Ligand Binding Modes and Rational Inhibitor Design for Kinase Drug Discovery(2008)157 cited
- → Discovery of a Potent, Selective, and Orally Active Proteasome Inhibitor for the Treatment of Cancer(2008)146 cited
- → High asymmetric induction during organometallic .beta.-addition to .alpha.,.beta.-ethylenic sulfoxides. Synthesis of optically active .beta.-alkylcarboxylic acids, .beta.-substituted cyclopentanones, and steroidal 11-oxoequilenin methyl ether(1981)129 cited
- CEP-7055: a novel, orally active pan inhibitor of vascular endothelial growth factor receptor tyrosine kinases with potent antiangiogenic activity and antitumor efficacy in preclinical models.(2003)
- → The Future of Antifungal Drug Therapy: Novel Compounds and Targets(2020)123 cited
- → Neurotrophic 3,9-Bis[(alkylthio)methyl]- and -Bis(alkoxymethyl)-K-252a Derivatives(1997)119 cited
- → Novel Peptidyl Phosphorus Derivatives as Inhibitors of Human Calpain I(1998)104 cited
- → Structure-guided identification of novel VEGFR-2 kinase inhibitors via solution phase parallel synthesis(2006)104 cited
- → Asymmetric induction during organometallic conjugate addition to enantiomerically pure 2-(arylsulfinyl)-2-cyclopentenones(1982)92 cited