Paul Eastwood
Almirall (Spain)(ES)
Publications by Year
Research Areas
Synthesis and Biological Evaluation, Asymmetric Synthesis and Catalysis, Synthetic Organic Chemistry Methods, Synthesis and Reactivity of Heterocycles, Phenothiazines and Benzothiazines Synthesis and Activities
Most-Cited Works
- → A versatile synthesis of 4-aryl tetrahydropyridines via palladium mediated Suzuki cross-coupling with cyclic vinyl boronates(2000)54 cited
- → Mapping the kinase domain of janus kinase 3(2003)50 cited
- → Total Synthesis of (+)-Dactylol via a Novel [3 + 5] Annulation Approach(1995)35 cited
- → Novel triazolopyridylbenzamides as potent and selective p38α inhibitors(2012)33 cited
- → Indolin-2-one p38α inhibitors III: Bioisosteric amide replacement(2011)33 cited
- → Identification of 2-Imidazopyridine and 2-Aminopyridone Purinones as Potent Pan-Janus Kinase (JAK) Inhibitors for the Inhaled Treatment of Respiratory Diseases(2019)32 cited
- → Structure based design of 4-(3-aminomethylphenyl)piperidinyl-1-amides: novel, potent, selective, and orally bioavailable inhibitors of βII tryptase(2005)29 cited
- → Indolin-2-one p38α inhibitors I: Design, profiling and crystallographic binding mode(2011)29 cited
- → [3 + 4] and [3 + 5] Annulation Reactions of .alpha.-(Phenylthio)Dicarbonyl Electrophiles with Bis(trimethylsilyl) Enol Ethers: Synthesis of Highly Functionalized Medium Ring Carbocycles(1995)28 cited
- → Chelation and Nonchelation Control in the [3 + 4] and [3 + 5] Annulation Reactions of Benzyloxy-Substituted Dicarbonyl Electrophiles with Bis(trimethylsilyl) Enol Ethers(1996)22 cited