Serge Pieters
Johnson & Johnson (United States)(US)Janssen (Belgium)(BE)Drug Discovery Laboratory (Norway)(NO)Janssen (United States)(US)
Publications by Year
Research Areas
Respiratory viral infections research, Hepatitis B Virus Studies, Immune Response and Inflammation, Chemical Synthesis and Analysis, Hepatitis C virus research
Most-Cited Works
- → 2-Amino-3,4-dihydroquinazolines as Inhibitors of BACE-1 (β-Site APP Cleaving Enzyme): Use of Structure Based Design to Convert a Micromolar Hit into a Nanomolar Lead(2007)145 cited
- → New 2-substituted 1,2,3,4-tetrahydrobenzofuro[3,2-c]pyridine having highly active and potent central α2-antagonistic activity as potential antidepressants(2000)69 cited
- → Design and Synthesis of a Novel Series of Bicyclic Heterocycles As Potent γ-Secretase Modulators(2012)60 cited
- → Synthesis and Pharmacological Characterization of Two Novel, Brain Penetrating P2X7 Antagonists(2013)46 cited
- → Novel Pyrimidine Toll-like Receptor 7 and 8 Dual Agonists to Treat Hepatitis B Virus(2016)40 cited
- → 2,4-Diaminoquinazolines as Dual Toll-like Receptor (TLR) 7/8 Modulators for the Treatment of Hepatitis B Virus(2018)26 cited